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Vosilasarm

Also known as: RAD-140, RAD140, Testolone, EP0062

Classification

Sarm

Regulatory Status

not-established

Overview

Vosilasarm (RAD-140, testolone) is a non-steroidal oral SARM that acts as an androgen receptor agonist; an investigational oncology program (EP0062) evaluates AR agonism in AR+/ER+ breast cancer, distinct from bodybuilding marketing.

Evidence and limitations

Human/preclinical evidence breakdown is not available in this record.

Pathways

androgen-receptor-signalingandrogen receptor agonismselective androgen receptor modulationandrogen receptor

Benefits

INN vosilasarm refers to RAD-140; early-phase oncology studies exist, but no FDA-approved indication, and bodybuilding uses are unapproved with hepatotoxicity case reports.

Interactions & cautions

other androgens, anabolic steroids, or SARMs — Additive androgenic and hepatotoxicity concerns (review)

hepatotoxic drugs or supplements — May worsen DILI risk (review)

These are observational flags for review, not individualized instructions.

Sources

Educational reference only — not medical advice.